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Inventor:

陈海军 (陈海军.) [1] (Scholars:陈海军) | 胡建达 (胡建达.) [2] | 陈策实 (陈策实.) [3] | 陈英玉 (陈英玉.) [4] | 刘蓉 (刘蓉.) [5] | 李财龙 (李财龙.) [6] | 高瑜 (高瑜.) [7] (Scholars:高瑜)

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incoPat

Abstract:

本发明属于医药技术领域,提供了一种哌嗪修饰的乌索酸衍生物及其制备方法和应用。以乌索酸为起始原料,经过四步反应制得哌嗪修饰的乌索酸衍生物:。该方法所用试剂为实验室常用试剂,且产物纯化方法较为简便,得到具有高抗肿瘤活性的哌嗪修饰的乌索酸衍生物。反应操作简单,易于处理,可以大量获得具有高生物活性的哌嗪修饰的乌索酸衍生物,以供医药研发的使用。

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Patent Info :

Type: 发明授权

Patent No.: CN201610229113.8

Filing Date: 2016/4/14

Publication Date: 2017/9/22

Pub. No.: CN105693815B

公开国别: CN

Applicants: 福州大学

Legal Status: 授权

Cited Count:

WoS CC Cited Count:

SCOPUS Cited Count:

ESI Highly Cited Papers on the List: 0 Unfold All

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Chinese Cited Count:

30 Days PV: 1

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