Divergent Synthesis of 1,1-Carbonyl Amino Alkyl Borons from Indoles - Details

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α-Boryl　carbonyl　species　and　α-boryl　amino　compounds　are　valuable　and　important　frameworks　in　organic　synthesis.　However,　the　strategies　that　could　merge　the　two　scaffolds　into　one　compound,　named　1,1-carbonyl　amino　alkyl　boron,　are　elusive　and　underdeveloped.　Herein,　we　present　an　efficient　method　that　could　address　this　gap　and　produce　1,1-carbonyl　amino　alkyl　borons　from　readily　accessible　indoles　via　oxidation　by　m-CPBA　or　oxone.　This　reaction　features　operational　simplicity,　divergent　synthesis,　broad　substrate　scope,　and　valuable　products.　　©　2023　American　Chemical　Society.

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[ 1 ] [Hou M.]Key Laboratory of Molecule Synthesis and Function Discovery, Fujian Province University, College of Chemistry, Fuzhou University, Fujian, Fuzhou, 350108, China
[ 2 ] [Wang Y.]Key Laboratory of Molecule Synthesis and Function Discovery, Fujian Province University, College of Chemistry, Fuzhou University, Fujian, Fuzhou, 350108, China
[ 3 ] [Li P.]Key Laboratory of Molecule Synthesis and Function Discovery, Fujian Province University, College of Chemistry, Fuzhou University, Fujian, Fuzhou, 350108, China
[ 4 ] [Ma X.]Key Laboratory of Molecule Synthesis and Function Discovery, Fujian Province University, College of Chemistry, Fuzhou University, Fujian, Fuzhou, 350108, China
[ 5 ] [Zhang G.]Key Laboratory of Molecule Synthesis and Function Discovery, Fujian Province University, College of Chemistry, Fuzhou University, Fujian, Fuzhou, 350108, China
[ 6 ] [Song Q.]Key Laboratory of Molecule Synthesis and Function Discovery, Fujian Province University, College of Chemistry, Fuzhou University, Fujian, Fuzhou, 350108, China
[ 7 ] [Song Q.]School of Chemistry and Chemical Engineering, Henan Normal University, Henan, Xinxiang, 453007, China

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Organic Letters

ISSN： 1523-7060

Year： 2023

Issue： 22

Volume： 25

Page： 4038-4043

4 . 9

JCR@2023

4 . 9 0 0

JCR@2023

ESI HC Threshold：39

JCR Journal Grade：1

CAS Journal Grade：1

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ESI Highly Cited Papers on the List： 0 Unfold All

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30 Days PV： 1

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