A Robust Copper-Catalyzed Cross-Coupling of Glycosyl Thiosulfonate and Boronic Acids Enables the Construction of Thioglycosides - Details

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An　efficient　and　stereoretentive　copper-catalyzed　cross-coupling　of　glycosyl　thiosulfonate　and　boronic　acid　for　the　construction　of　thioglycosides　is　described.　The　good　functional　group　compatibility　of　this　method　allows　the　preparation　of　many　bioactive　aryl/alkenyl　thioglycosides,　including　the　hSGLT1　inhibitor.　©　2023　American　Chemical　Society

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[ 1 ] [Sun Z.]Institute of Pharmaceutical Science and Technology, College of Chemistry, Fuzhou University, Fuzhou, 350108, China
[ 2 ] [Sun Z.]Qingyuan Innovation Laboratory, Quanzhou, 362801, China
[ 3 ] [Yan W.]Institute of Pharmaceutical Science and Technology, College of Chemistry, Fuzhou University, Fuzhou, 350108, China
[ 4 ] [Xie L.]Institute of Pharmaceutical Science and Technology, College of Chemistry, Fuzhou University, Fuzhou, 350108, China
[ 5 ] [Liu W.]Institute of Pharmaceutical Science and Technology, College of Chemistry, Fuzhou University, Fuzhou, 350108, China
[ 6 ] [Xu C.]Institute of Pharmaceutical Science and Technology, College of Chemistry, Fuzhou University, Fuzhou, 350108, China
[ 7 ] [Xu C.]Key Laboratory of Organofluorine Chemistry, Shanghai Institute of Organic Chemistry, CAS, Shanghai, 200032, China
[ 8 ] [Chen F.-E.]Institute of Pharmaceutical Science and Technology, College of Chemistry, Fuzhou University, Fuzhou, 350108, China
[ 9 ] [Chen F.-E.]Qingyuan Innovation Laboratory, Quanzhou, 362801, China
[ 10 ] [Chen F.-E.]Engineering Center of Catalysis and Synthesis for Chiral Molecules, Department of Chemistry, Fudan University, Shanghai, 200433, China
[ 11 ] [Chen F.-E.]Shanghai Engineering Center of Industrial Asymmetric Catalysis for Chiral Drugs, Fudan University, Shanghai, 200433, China

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Organic Letters

ISSN： 1523-7060

Year： 2023

Issue： 31

Volume： 25

Page： 5714-5718

4 . 9

JCR@2023

4 . 9 0 0

JCR@2023

ESI HC Threshold：39

JCR Journal Grade：1

CAS Journal Grade：1

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ESI Highly Cited Papers on the List： 0 Unfold All

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30 Days PV： 1

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